Triptorelin Pamoate
4144950
Bachem Regulatory Documentation
DMF
Synonyms
(D-Trp6)-LHRH; Triptorelin Embonate
Sequence
Pyr-His-Trp-Ser-Tyr-D-Trp-Leu-Arg-Pro-Gly-NH2 pamoate salt
Fields of Application
Active Substance
Triptorelin Pamoate (also called Triptorelin Embonate) is a potent LHRH (GnRH) agonist. Triptorelin Pamoate is a salt form of triptorelin suitable for obtaining controlled release formulations. After a transient increase, continuous administration of triptorelin results in downregulation of LH and FSH levels followed by a suppression of ovarian and testicular steroid biosynthesis.
Molecular Information
Molecular Formula
C64H82N18O13
Relative Molecular Mass
1311.47 g/mol
CAS-Number
57773-63-4 (net), 124508-66-3 (pamoate)
Long-term Storage
-20 ± 5°C